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Search Results for " estrogen receptor/err "

20

Compounds

Cat No. Product Name Synonyms Targets
T4388 PHTPP Estrogen Receptor/ERR , Estrogen/progestogen Receptor
PHTPP is a selective ERβ antagonist.
TN1052 Lindleyin Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Lindleyin is a novel phytoestrogen and might trigger many of the biological responses evoked by the physiological estrogens.
T15249 Estrogen receptor modulator 1 Estrogen Receptor/ERR
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.4...
T13768 (+)-Medicarpin Estrogen/progestogen Receptor
(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymiscium yucatamun, Machaerium aristulatum, and Platymiscium flo...
T5S0543 Isocurcumenol Apoptosis , Estrogen Receptor/ERR , Reductase
1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).
T3665 Tectoridin Shekanin Estrogen Receptor/ERR , Reductase
Tectoridin (Shekanin) possesses an estrogenic and thyroid hormone-like agent by activating estrogen and thyroid hormone receptors. Tectoridin has anti-oxidant, anti-inflammatory and hypoglycemic activities; Tectoridin an...
T3855 Tracheloside Estrogen Receptor/ERR , Phosphorylase
Tracheloside significantly decreases the activity of alkaline phosphatase (IC50: 0.31 μg/ml), a level of inhibition comparable to that of tamoxifen (IC50: 0.43 μg/ml).
T16566 Propyl pyrazole triol PPT Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 410 times higher compared with estrogen receptor beta (ERβ: ...
T7904 SR 19881 Estrogen/progestogen Receptor
SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding assay and an EC50 value of 4.7 μM in a cell-based assay).
T8984 FLTX1 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under permeabilized and non-permeabilized conditions. Additionally,...
T0593 XCT790 Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Autophagy
XCT790 is a potent, selective and inverse agonist of estrogen-related receptor alpha(ERRα).
TQ0295 Coumestrol Estrogen Receptor/ERR
Coumestrol that existed in soybean products suppresses the proliferation of ES2 cells (IC50: 50 μM). It exhibits activities against neurological disorders, cancers and autoimmune diseases.
T15364 G-1 Estrogen Receptor/ERR , GPR
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
T7389 G15 Estrogen Receptor/ERR
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
T14987 CMP8 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, res...
T5531 GSK-4716 Estrogen Receptor/ERR
GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand
T3975 AZD9496 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.
T3958 WAY-200070 WAY 200070 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).
T13542 α-Zearalenol Estrogen Receptor/ERR
α-Zearalenol is one of the major metabolites of Zearalenone. α-Zearalenol has structural analogy to estrogen, thus α-Zearalenol can bind to estrogen receptors (ERs).
T1216 Diethylstilbestrol Stilbestrol,DES Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Diethylstilbestrol (DES) is used in the treatment of menopausal and postmenopausal disorders.

Compounds

PHTPP
T4388
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Lindleyin
TN1052
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Estrogen receptor modulator 1
T15249
Synonym:
Target: Estrogen Receptor/ERR
(+)-Medicarpin
T13768
Synonym:
Target: Estrogen/progestogen Receptor
Isocurcumenol
T5S0543
Synonym:
Target: Apoptosis, Estrogen Receptor/ERR, Reductase
Tectoridin
T3665
Synonym: Shekanin
Target: Estrogen Receptor/ERR, Reductase
Tracheloside
T3855
Synonym:
Target: Estrogen Receptor/ERR, Phosphorylase
Propyl pyrazole triol
T16566
Synonym: PPT
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
SR 19881
T7904
Synonym:
Target: Estrogen/progestogen Receptor
FLTX1
T8984
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
XCT790
T0593
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Autophagy
Coumestrol
TQ0295
Synonym:
Target: Estrogen Receptor/ERR
G-1
T15364
Synonym:
Target: Estrogen Receptor/ERR, GPR
G15
T7389
Synonym:
Target: Estrogen Receptor/ERR
CMP8
T14987
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
GSK-4716
T5531
Synonym:
Target: Estrogen Receptor/ERR
AZD9496
T3975
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
WAY-200070
T3958
Synonym: WAY 200070
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
α-Zearalenol
T13542
Synonym:
Target: Estrogen Receptor/ERR
Diethylstilbestrol
T1216
Synonym: Stilbestrol,DES
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
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TargetMol